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承师创新3

李正名简历3

李正名自述5

饮水思源——恩师杨石先先生对农药化学学科的重要贡献及其学术思想9

业绩与奖项16

主要科研项目18

论文选登23

1957年23

萘和苯的衍生物类生长素对植物插枝生根作用的初步报告23

1959年35

有机磷杀虫剂的研究Ⅰ35

1962年44

有机磷杀虫剂的研究Ⅱ44

1963年48

有机磷杀虫剂的研究Ⅲ48

1965年54

有机磷杀虫剂的研究Ⅶ54

1983年63

UV-Ozonation and Land Disposal of Aqueous Pesticide Wastes63

内吸杀菌剂三唑醇立体异构体研究初报69

1984年73

棉铃虫拟信息素正十四烷基甲酸酯及有关化合物的触角电位反应73

A Convenient Synthetic Route for the Sex Pheromone of the Asian Corn Borer Moth（Ostrinia furnacalis Guenee）76

1987年83

内吸性杀菌剂三唑醇（酮）立体异构体的研究（Ⅱ）83

1-（4-氯苯氧基-3，3-二甲基-1-（1，2，4-三氮唑-1基）-丁醇2右旋A体的晶体结构和绝对构型89

1989年93

A Stereoselective Synthesis of Pear Ester via Arsenic Ylide93

1990年96

The Chemical Characterization of the Cephalic Secretion of the Australian Colletid Bee，Hylaeus albonitens（Gnathoprosopls Cockerell）96

The Wittig Sigmatropic Rearrangement in a Conjugated Diene System Ⅰ105

山梨酸的合成及其生物活性研究111

1991年120

茶尺蠖性信息素化学结构研究初报120

1992年123

新磺酰脲类化合物的合成、结构及构效关系研究（Ⅰ）123

1993年129

新磺酰脲类化合物的合成、结构及构效关系研究（Ⅱ）129

Structural Elucidation of Sex Pheromone Components of the Geometridae Semiothisa cinerearia（Bremer et Grey）in China134

1994年140

新磺酰脲类化合物的合成、结构及构效关系研究（Ⅲ）140

The Reaction of α-oxo-α-Triazolylketene Dithioacetal with Amines，Hydrazine and Guanidine144

Studies on Sex Pheromone of Ectropis obliqua Prout147

1995年155

Synthesis of 5-Mercaptoalkylamino-and 5-Anilinoalkylthiopyrazolyl-1，2，4-Triazoles by Ring Chain Transformation155

1996年161

Synthesis and base-catalyzed Protodesilylation of 5-（Silylmethylthio）-3（2H）-Pyridazinone Derivatives161

Synthesis of 5-mercaptoalkylthiopyrazolyl-and3-mercaptoalkyl thioisoxazolyl-1，2，4-triazoles by Ring Chain Transformation168

1997年172

新磺酰脲类化合物的合成、结构及构效关系研究（Ⅴ）172

新型杀菌剂β-甲氧基丙烯酸甲酯类化合物的合成方法概述176

1998年182

3-吡唑基-6-取代均三唑并［3，4-b］-1，3，4-噻二唑的合成及生物活性182

Syntheses of Di-heterocyclic Compounds；Pyrazolylimidazoles and Isoxazolylimidazoles187

3-芳基磺酰氧基（取代）异噻唑的合成及除草活性192

应用CoMFA研究磺酰脲类化合物的三维构效关系197

2，5-二吡唑基-1，3，4-噁二唑的一锅煮法合成及生物活性202

1999年205

2-芳甲酰氨基硫羰基-3-异噻唑酮及4-氰基-5-甲硫基-2-芳甲酰氨基硫羰基-3-异噻唑酮的合成与生物活性205

The Design and Synthesis of ALS Inhibitors from Pharmacophore Models210

2000年215

新磺酰脲类化合物的合成、结构及构效关系研究（Ⅵ）215

Synthesis and Fungicidal Activity against Rhizoctonia solani of 2-Alkyl（Alkylthio）-5-pyrazolyl-1，3，4-oxadiazoles（Thiadiazoles）220

2001年229

N-（取代嘧啶-2′-基）-2-三氟乙酰氨基苯磺酰脲的合成及除草活性229

新磺酰脲类除草活性构效关系的研究233

2002年240

卤代-2-（3-甲基-5-取代-4H-1，2，4-三唑-4-基）-苯甲酸的合成240

5-依维菌素B1a酯的合成和生物活性244

2-（1H-咪唑-1-基）-1-（2，3，4-三甲氧基）苯乙酮肟酯新化合物合成与生物活性研究256

2003年262

1，3-二甲基-5-甲硫基-4-苯腙基羰基吡唑的合成及抑菌活性262

Metal Ion Interactions with Sugars.The Crystal Structure and FT-IR Study of the NdCl3-ribose Complex266

3-Methylthio-pyrano［4，3-c］pyrazol-4（2H）-ones from 3-（Bis-methylthio）methylene-2H-pyran-2，4-diones and Hydrazines277

2004年281

新单取代苯磺酰脲衍生物的合成及生物活性281

N-（4-取代嘧啶-2-基）苄基磺酰脲和苯氧基磺酰脲的3D-QSAR研究287

基于酮醇酸还原异构酶KARI复合物晶体结构的三维数据库搜寻291

N-杂环-3-N′-苄氧羰基-β-氨基丁酰胺的合成和结构表征296

Synthesis and Biological Activity of Novel 2-Methyl-4-trifluoromethyl-thiazole-5-carboxamide derivatives302

Metal-ion Interactions with Sugars Crystal Structures and FT-IR Studies of the LaCl3-ribopyranose and CeCl3-ribopyranose Complexes308

2005年324

一类新型嘧啶苯氧（硫）醚的合成及生物活性324

4-（取代嘧啶-2-基）-1-芳磺酰基氨基脲化合物的合成与表征331

Synthesis and Fungicidal Activity of Novel 2-Oxocycloalkylsulfonylureas339

Synthesis，Crystal Structure and Herbicidal Activity of Mimics of Intermediates of the KARI Reaction349

Synthesis and Herbicidal Activity of 2-Alkyl（aryl）-3-methylsulfonyl（sulfinyl）pyrano-［4，3-c］pyrazol-4（2H）-ones358

2006年364

单嘧磺隆除草剂的晶体构象-活性构象转换的密度泛函理论研究364

O-取代苯基-O-（2-硬脂酰胺基）乙基-N，N-二（2-氯乙基）磷酰胺的合成和生物活性376

3-N-苄氧羰基-β-氨基丁酸水杨酸酯类化合物的合成及其生物活性383

Synthesis and Crystal Structure of 5-N-i-Propyl-2-（2′-nitrobenzene-sulfonyl）-glutamine389

Synthesis，Dimeric Crystal Structure，and Biological Activities of N-（4-Methyl-6-oxo-1，6-dinydro-pyrimidin-2-yl）-N′-（2-trifluoro-methyl-phenyl）-guanidine394

Microwave and Ultrasound Irradiation-Assisted Synthesis of Novel Disaccharide-Derived Arylsulfonyl Thiosemicarbazides400

2007年406

Synthesis of New Plant Growth Regulator：N-（fatty acid）O-aryloxyacetyl Ethanolamine406

Synthesis，Bioactivity，Theoretical and Molecular Docking Study of 1-Cyano-N-substituted-cyclopropanecarboxamide as Ketol-acid Reductoisomerase Inhibitor411

单嘧磺隆晶体-活性构象转换的分子动力学模拟420

基于受体结构的AHAS抑制剂的设计、合成及生物活性427

The Design，Synthesis，and Biological Evaluation of Novel Substituted Purines as HIV-1 Tat-TAR Inhibitors431

酵母AHAS酶与磺酰脲类抑制剂作用模型的分子对接研究444

2008年450

High Throughput Screening Under Zinc-Database and Synthesis a Dialkylphos-phinic Acid as a Potential Kari Inhibitor450

N-（4′-取代嘧啶-2′-基）-2-甲氧羰基-5-（取代）苯甲酰胺基苯磺酰脲化合物的合成及除草活性研究453

Synthesis and Herbicidal Activity of Novel Sulfonylureas Containing Thiadiazol Moiety465

The Outset Innovation of Agrochemicals in China471

2009年477

Quantitive-structure Activity Relationship（QSAR）Study of a New Heterocyclic Insecticides Using CoMFA and CoMSIA477

Design，Synthesis，and Fungicidal Activity of Novel Analogues of Pyrrolnitrin483

新型苯环5-（取代）苯甲酰胺基苯磺酰脲类化合物的比较定量构效关系研究496

Regioselective Synthesis of Novel 3-Alkoxy（phenyl）thiophosphorylamido-2-（per-O-acetylglycosyl-1′-imino） Thiazolidine-4-one Derivatives from O-alkyl N4-glycosyl（thiosemicarbazido） Phosphonothioates501

Synthesis，Herbicidal Activities and Comparative Molecular Field Analysis Study of Some Novel Triazolinone Derivatives512

Synthesis，Antifungal Activities and 31D-QSAR Study of N-（5-substituted-1，3，4-thiadiazol-2-yl） Cyclopropanecarboxamides526

Synthesis，Bioactivity and SAR Study of N′-（5-substituted-1，3，4-thiadiazol-2-yl）-N-cyclopropylformyl-thioureas as Ketol-acidReductoisomerase Inhibitors535

Synthesis and Biological Activity of Novel 2，3-Dihydro-2-phenylsulfonyl-hydrazono-3-（2′，3′，4′，6′-tetra-O-acetyl-β-D-glucopyranosyl）thiazoles546

4，5，6-三取代嘧啶苯磺酰脲类化合物的生物活性、分子对接与3D-QSAR关系研究552

2010年559

Synthesis， Crystal Structure and Insecticidal Activities of Novel Neonicotinoid Derivatives559

区域选择性合成2-取代磺酰基亚肼基-3-全乙酰糖基-2， 3-二氢噻唑及其表征、生物活性研究567

3位苯甲酰腙和亚氨基取代硫脲取代的吲哚满二酮衍生物的合成及对AHAS的抑制活性573

Synthesis and Biological Activity of Some Novel Trifluoromethyl-Substituted 1，2，4-Triazole and Bis（1，2，4-Triazole） Mannich Bases Containing Piperazine Rings578

Synthesis and Fungicidal Activity of Novel Aminophenazine-1-carboxylate Derivatives594

High Throughput Receptor-based Virtual Screening under ZINC Database，Synthesis，and Biological Evaluation of Ketol-acid Reductoisomerase Inhibitors618

2011年627

Synthesis and Insecticidal Activities of Novel Analogues of Chlorantraniliprole Containing Nitro Group627

Modulations of High-voltage Activated Ca2+ Channels in the Central Neurones of Spodoptera Exigua by Chlorantraniliprole634

Synthesis，Structure and Biological Activity of Novel 1，2，4-Triazole Mannich Bases Containing a Substituted Benzylpiperazine Moiety641

Design，Synthesis and Antifungal Activities of Novel Pyrrole Alkaloid Analogs654

Synthesis and Insecticidal Evaluation of Novel N-Pyridylpyrazolecarboxamides Containing Different Substituents in the ortho-Position675

Synthesis，Crystal Structure，Bioactivity and DFT Calculation of New Oxime Ester Derivatives Containing Cyclopropane Moiety684

2012年693

The Structure-activity Relationship in Herbicidal Monosubstituted Sulfonylureas693

Synthesis，Crystal Structure and Biological Activities of Novel Anthranilic （ Isoph-thalic）Acid Esters708

Synthesis and Evaluation of Novel Monosubstituted Sulfonylurea Derivatives as Antituberculosis Agents716

基于Ugi反应的新型鱼尼丁受体杀虫剂的设计、合成及生物活性736

Synthesis and Insecticidal Activities of Novel Anthranilic Diamides Containing Acylthiourea and Acylurea746

Design，Synthesis and Biological Activities of Novel Anthranilic Diamide Insecticide Containing Trifluoroethyl Ether760

Evaluation of the in Vitro and Intracellular Effiicacy of New Monosubstituted Sulfonylureas against Extensively Drug-resistant Tuberculosis779

2013年786

Synthesis and Insecticidal Evaluation of Novel N-Pyridylpyrazolecarboxamides Containing Cyano Substituent in the ortho-Position786

N-［4-氯-2-取代氨基甲酰基-6-甲基苯基］-1-芳基-5-氯-3-三氟甲基-1 H-吡唑-4-甲酰胺的合成及生物活性795

Synthesis，Insecticidal Activities，and SAR Studies of Novel Pyridylpyrazole Acid Derivatives Based on Amide Bridge Modification of Anthranilic Diamide Insecticides805

Design，Synthesis and Structure-activity of N-Glycosyl-1-pyridyl-1H- pyrazole-5-carboxamide as Inhibitors of Calcium Channels826

新型含三唑啉酮的磺酰脲类化合物的合成、晶体结构及除草活性研究839

Design，Syntheses and Biological Activities of Novel Anthranilic Diamide Insecticides Containing N-Pyridylpyrazole853

Synthesis and Biological Activities of Novel Anthranilic Diamides Analogues Containing Benzo［b］thiophene865

附录879

附录1论文总目录879

附录2专利及著作目录911

附录3历年指导的学生名单915